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GPR54 (Kiss1R) is a rhodosin‑family GPCR receptor that binds kisspeptin‑10. It governs puberty onset and reproductive hormone secretion, and participates in energy metabolism regulation. The kisspeptin‑10/GPR54 axis drives intracellular Gq‑mediated signaling, and represents a key therapeutic target for reproductive‑related drug research. Our GPR54(Kiss1R) stable CHO cell lines have been validated in HTRF IP‑One assays to support your drug discovery programs.